5-HT Receptor Inhibitors

5-HT₁ Receptor

5-HT₂ Receptor

5-HT₃ Receptor

5-HT₄ Receptor

5-HT₅ Receptor

5-HT₆ Receptor

5-HT₇ Receptor

5-HT Receptor

5-HT Receptor Inhibitors, Agonists, Antagonists, Activators & Modulators

Product Name	5-HT₁ Receptor	5-HT₂ Receptor	5-HT₃ Receptor	5-HT₄ Receptor	5-HT₅ Receptor	5-HT₆ Receptor	5-HT₇ Receptor	5-HT Receptor	Purity
Serotonin hydrochloride								serotonin	99.97%
SCH-23390 hydrochloride		5-HT_2C Receptor, Ki: 9.3 nM							99.91%
Puerarin		5-HT_2C Receptor							99.42%
Tianeptine sodium salt								serotonin	99.90%
Tianeptine								serotonin	99.84%
MT-1207		5-HT_2A Receptor, IC₅₀: 0.27 nM 5-HT_2A Receptor, Ki: 0.079 nM							99.96%
Harmine		5-HT_2A Receptor, Ki: 397 nM							99.88%
Clozapine		5-HT_2A Receptor, Ki: 4 nM (Inhibitor)							99.97%
Scopolamine hydrobromide			5-HT₃ Receptor, IC₅₀: 2.09 μM						99.93%
Scopolamine			5-HT₃ Receptor, IC₅₀: 2.09 μM						99.86%
Olanzapine	5-HT₁ Receptor, Ki: 7 nM	5-HT_2A Receptor, Ki: 4 nM 5-HT_2C Receptor, Ki: 11 nM	5-HT₃ Receptor, Ki: 57 nM			5-HT₆ Receptor, Ki: 5 nM			99.83%
Risperidone		5-HT_2A Receptor, Ki: 4.8 nM							99.92%
Vortioxetine			5-HT_3A Receptor, Ki: 3.7 nM				Human 5-HT₇ Receptor , Ki: 19 nM		99.81%
Aripiprazole	5-HT_1A Receptor, Ki: 4.2 nM								99.95%
Ondansetron			5-HT₃ Receptor						99.37%
GTS-21 dihydrochloride			5-HT_3A Receptor, IC₅₀: 3.1 μM						99.92%
Vortioxetine hydrobromide			5-HT_3A Receptor, Ki: 3.7 nM				5-HT₇ Receptor, Ki: 19 nM		99.91%
Thioridazine hydrochloride								serotonin	99.96%
Volinanserin		5-HT₂ Receptor, Ki: 0.36 nM							99.76%
Vilazodone Hydrochloride	5-HT_1A Receptor								99.94%
Amitriptyline hydrochloride	5-HT_1A Receptor, IC₅₀: 450 nM 5-HT_1B Receptor, IC₅₀: 40 nM	5-HT_2A Receptor, IC₅₀: 4 nM 5-HT_2B Receptor, IC₅₀: 40 nM 5-HT_2C Receptor, IC₅₀: 6 nM							98.91%
BW-723C86		5-HT_2B Receptor							99.80%
SB-269970 hydrochloride							5-HT₇ Receptor, pKi: 8.3		98.62%
WAY-100635	5-HT_1A Receptor, pIC₅₀: 8.87 5-HT_1A Receptor, pA2: 9.71								99.44%
Pimavanserin		5-HT_2A Receptor, pIC₅₀: 8.7							99.86%
PCPA methyl ester hydrochloride								serotonin	99.89%
Ketanserin		5-HT₂ Receptor							99.89%
Brexpiprazole	5-HT_1A Receptor, Ki: 0.12 nM	5-HT_2A Receptor, Ki: 0.47 nM							99.85%
Cisapride				5-HT₄ Receptor, EC₅₀: 0.14 μM					99.72%
Vilazodone	5-HT_1A Receptor								99.84%
SEP-363856 hydrochloride	5-HT_1A Receptor, EC₅₀: 2.3 μM 5-HT_1B Receptor, EC₅₀: 15.6 μM 5-HT_1D Receptor, EC₅₀: 0.262 μM	5-HT_2A Receptor, EC₅₀: >10 μM 5-HT_2C Receptor, EC₅₀: 30 μM					5-HT₇ Receptor, EC₅₀: 6.7 μM		99.57%
8-OH-DPAT	5-HT_1A Receptor, pIC₅₀: 8.19						5-HT₇ Receptor, Ki: 466 nM		99.26%
Pindolol	5-HT_1A Receptor								99.91%
Quetiapine	5-HT_1A Receptor, pKi: 5.74 5-HT_1A Receptor, pEC₅₀: 4.77	5-HT_2A Receptor, pKi: 7.54 5-HT_2C Receptor, pKi: 5.55							99.88%
Tegaserod maleate		5-HT_2B Receptor (Antagonist)		5-HT₄ Receptor (Agonist)					99.93%
DOI hydrochloride		Human 5-HT_2A Receptor, Ki: 0.7 nM Human 5-HT_2C Receptor, Ki: 2.4 nM human 5-HT_2B Receptor, Ki: 20 nM							99.61%
Perphenazine	5-HT_1A Receptor, Ki: 421 nM	5-HT_2A Receptor, Ki: 5.6 nM				5-HT₆ Receptor, Ki: 17 nM	5-HT₇ Receptor, Ki: 23 nM		99.95%
Prucalopride				5-HT_4A Receptor, pKi: 8.6 5-HT_4B Receptor, pKi: 8.1					99.81%
SB 242084		5-HT_2C Receptor, pKi: 9.0							99.88%
Lurasidone	5-HT_1A Receptor, IC₅₀: 6.75 nM						5-HT₇ Receptor, IC₅₀: 0.495 nM		99.49%
Ritanserin		5-HT₂ Receptor, IC₅₀: 0.9 nM							99.68%
Nuciferine	5-HT_1A Receptor, EC₅₀: 3.2 μM	5-HT_2C Receptor, IC₅₀: 131 nM 5-HT_2A Receptor, IC₅₀: 478 nM 5-HT_2B Receptor, IC₅₀: 1 μM				5-HT₆ Receptor, EC₅₀: 700 nM	5-HT₇ Receptor, IC₅₀: 150 nM		99.46%
Cariprazine	5-HT_1A Receptor, Ki: 2.6 nM								99.83%
Agomelatine		5-HT_2C Receptor, pKi: 6.4 (native porcine) 5-HT_2C Receptor, pKi: 6.2 (human)							99.88%
GR 113808	5-HT_1A Receptor	5-HT_2A Receptor 5-HT_2C Receptor	5-HT₃ Receptor	5-HT₄ Receptor					99.96%
Cariprazine hydrochloride	5-HT_1A Receptor, Ki: 2.6 nM								99.90%
Paliperidone		5-HT_2A Receptor							99.69%
Ziprasidone	Rat 5-HT_1A Receptor, Ki: 3.4 nM human 5-HT_1A Receptor, Ki: 2.5 nM	Rat 5-HT_2A, Ki: 0.42 nM							99.81%
Alosetron Hydrochloride			5-HT₃ Receptor						99.76%
8-OH-DPAT hydrobromide	5-HT_1A Receptor, pIC₅₀: 8.19								99.89%
Alprenolol	5-HT_1A Receptor								99.94%
SB 204741		human 5-HT_2B Receptor, pKi: 7.1							99.85%
Ketanserin tartrate		5-HT₂ Receptor							99.99%
Sumatriptan succinate	5-HT_1D Receptor, Ki: 17 nM 5-HT_1B Receptor, Ki: 27 nM 5-HT_1A Receptor, Ki: 100 nM 5-HT_1D Receptor, IC₅₀: 7.3 nM 5-HT_1B Receptor, IC₅₀: 9.3 nM 5-HT_1F Receptor, IC₅₀: 17.8 nM								99.94%
Metergoline		5-HT_2A Receptor, pKi: 8.64 5-HT_2B Receptor, pKi: 8.75 5-HT_2C Receptor, pKi: 8.75					Human 5-HT₇ Receptor , Ki: 16 nM		99.89%
Mirtazapine		5-HT₂ Receptor, pKi: 8.05	5-HT₃ Receptor, pKi: 8.1						99.94%
Rotigotine	5-HT_1A Receptor, Ki: 30 nM						5-HT₇ Receptor, Ki: 86 nM		99.99%
Gamma-Mangostin		5-HT_2A Receptor							99.91%
Methiothepin mesylate	5-HT_1A Receptor, pKd: 7.10 5-HT_1B Receptor, pKd: 7.28 5-HT_1C Receptor, pKd: 7.56 5-HT_1D Receptor, pKd: 6.99	5-HT_2A Receptor, pKi: 8.50 5-HT_2B Receptor, pKi: 8.68 5-HT_2C Receptor, pKi: 8.35			5-HT_5A Receptor, pKd: 7.0 5-HT_5B Receptor, pKd: 7.8	5-HT₆ Receptor, pKd: 8.74	5-HT₇ Receptor, pKd: 8.99		99.60%
Alprenolol hydrochloride	5-HT_1A Receptor								99.76%
SB-224289 hydrochloride	5-HT_1B Receptor								≥99.0%
Loxapine		human 5-HT₂							99.69%
Sumatriptan	5-HT_1A Receptor, Ki: 100 nM 5-HT_1B Receptor, Ki: 27 nM 5-HT_1D Receptor, Ki: 17 nM 5-HT_1D Receptor, IC₅₀: 7.3 nM 5-HT_1B Receptor, IC₅₀: 9.3 nM 5-HT_1F Receptor, IC₅₀: 17.8 nM								99.90%
R 59-022								serotonin	99.82%
Asenapine maleate		5-HT_2A Receptor, Ki: 0.06 nM 5-HT_2C Receptor, Ki: 0.03 nM					5-HT₇ Receptor, Ki: 0.13 nM		99.95%
Nefazodone hydrochloride		5-HT_2A Receptor, Ki: 5.8 nM							99.87%
Sertindole		5-HT_2A Receptor 5-HT_2C Receptor							99.92%
Loxapine succinate		human 5-HT₂							99.81%
Tegaserod				5-HT₄ Receptor					99.89%
Eucalyptol			5-HT₃ Receptor						≥98.0%
Prucalopride succinate				5-HT_4A Receptor, pKi: 8.6 5-HT_4B Receptor, pKi: 8.1					99.95%
Cefaclor								5-HT Receptor	99.61%
RS-127445 hydrochloride		5-HT_2A Receptor, pKi: 6.3 5-HT_2C Receptor, pKi: 6.4 5-HT_2B Receptor, pKi: 9.5	5-HT₃ Receptor, pKi: <6		5-HT₅ Receptor, pKi: <6	5-HT₆ Receptor, pKi: <6			99.78%
Palonosetron hydrochloride			5-HT₃ Receptor						99.96%
Rotigotine Hydrochloride	5-HT_1A Receptor, Ki: 30 nM						5-HT₇ Receptor, Ki: 86 nM		99.65%
Trimipramine maleate		5-HT₂ Receptor, pKi: 8.10							99.82%
SKF-83566		5-HT₂ Receptor, Ki: 11 nM							99.86%
Rotundine	5-HT_1A Receptor, IC₅₀: 370 nM								99.96%
LP-211	5-HT_1A Receptor, Ki: 188 nM						5-HT₇ Receptor, Ki: 0.58 nM		99.61%
Pimavanserin hemitartrate		5-HT_2A Receptor, pIC₅₀: 8.73 5-HT_2A Receptor, pKi: 9.3							99.91%
Cyproheptadine hydrochloride		5-HT₂ Receptor							99.94%
Roluperidone		5-HT_2A Receptor, Ki: 7.53 nM							99.86%
Tandospirone	5-HT_1A Receptor, Ki: 27 nM								99.41%
Lumateperone tosylate		5-HT_2A Receptor, Ki: 0.54 nM							99.53%
Gepirone	5-HT_1A Receptor								99.88%
NAS-181 dimesylate	Rat 5-HT_1B Receptor, IC₅₀: 47 nM								98.44%
SB-699551					5-HT_5A Receptor, pKi: 8.3				99.53%
UNC9994 hydrochloride	5-HT_1A Receptor, Ki: 26 nM	5-HT_2A Receptor, Ki: 140 nM 5-HT_2B Receptor, Ki: 25 nM 5-HT_2C Receptor, Ki: 512 nM							98.83%
Blonanserin		5-HT_2A Receptor, Ki: 0.812 nM 5-HT_2C Receptor, Ki: 26.4 nM				5-HT₆ Receptor, Ki: 11.7 nM			99.62%
Ondansetron hydrochloride dihydrate			5-HT₃ Receptor						99.94%
Mosapride citrate				5-HT₄ Receptor					99.96%
Metoclopramide			5-HT₃ Receptor, IC₅₀: 308 nM						99.94%
Sarpogrelate hydrochloride		5-HT_2A Receptor, pKi: 8.52 5-HT_2B Receptor, pKi: 6.57 5-HT_2C Receptor, pKi: 7.43							99.09%
SB-277011 hydrochloride	5-HT_1D Receptor 5-HT_1B Receptor								98.54%
Eletriptan hydrobromide	5-HT_1B Receptor, Ki: 0.92 nM 5-HT_1D Receptor, Ki: 3.14 nM								99.81%
Piboserod				5-HT₄ Receptor					99.09%
Granisetron Hydrochloride			5-HT₃ Receptor, IC₅₀: 17 μM						99.87%
Setiptiline maleate		5-HT_2A Receptor 5-HT_2C Receptor	5-HT₃ Receptor						99.94%
Ansofaxine hydrochloride								serotonin, IC₅₀: 723 nM	99.72%
(Z)-Thiothixene								serotonin	99.84%
2-Methyl-5-HT			5-HT₃ Receptor						98.73%
Syk Inhibitor II								serotonin, IC₅₀: 460 nM	98.05%
Lurasidone Hydrochloride	5-HT_1A Receptor, IC₅₀: 6.75 nM						5-HT₇ Receptor, IC₅₀: 0.495 nM		99.96%
Quetiapine hemifumarate	5-HT_1A Receptor, pKi: 5.74 5-HT_1A Receptor, pEC₅₀: 4.77	5-HT_2A Receptor, pKi: 7.54 5-HT_2C Receptor, pKi: 5.55							99.94%
Buspirone	5-HT_1A Receptor								99.86%
Harmine hydrochloride		5-HT_2A Receptor, Ki: 397 nM							99.93%
Paliperidone palmitate		5-HT_2A Receptor							98.41%
Asenapine	5-HT_1B Receptor, pKi: 8.4 5-HT_1A Receptor, pKi: 8.6	5-HT_2A Receptor, pKi: 10.2 5-HT_2C Receptor, pKi: 10.5 5-HT_2B Receptor, pKi: 9.8			5-HT₅ Receptor, pKi: 8.8	5-HT₆ Receptor, pKi: 9.6	5-HT₇ Receptor, pKi: 9.9		99.62%
5-Methoxytryptamine	5-HT₁ Receptor	5-HT₂ Receptor		5-HT₄ Receptor	5-HT₅ Receptor	5-HT₆ Receptor	5-HT₇ Receptor		99.91%
Granisetron			5-HT₃ Receptor, IC₅₀: 17 μM						99.95%
Norfluoxetine hydrochloride								5-HT Receptor	99.58%
Talipexole dihydrochloride			5-HT₃ Receptor						99.80%
Ziprasidone hydrochloride monohydrate	Rat 5-HT_1A Receptor, Ki: 3.4 nM	Rat 5-HT_2A, Ki: 0.42 nM							99.74%
S1RA		human 5-HT_2B Receptor, Ki: 328 nM							99.43%
Sarizotan	5-HT_1D Receptor, IC₅₀: 500 nM (calf) 5-HT_1B Receptor, IC₅₀: 600 nM (rat) 5-HT_1A Receptor, IC₅₀: 6.5 nM (rat) 5-HT_1A Receptor, IC₅₀: 0.1 nM (human)	5-HT_2A Receptor, IC₅₀: 960 nM (rat, agonist site) 5-HT_2A Receptor, IC₅₀: 587 nM (human, antagonist site) 5-HT_2C Receptor, IC₅₀: 800 nM (pig) 5-HT_2B Receptor, IC₅₀: 108 nM (human)	5-HT₃ Receptor, IC₅₀: 3500 nM (NG 108 cells)		5-HT_5A Receptor, IC₅₀: 313 nM (human)	5-HT₆ Receptor, IC₅₀: 3300 nM (human)	5-HT₇ Receptor, IC₅₀: 10 nM (human)		98.74%
AS19	5-HT_1A Receptor, Ki: 89.7 nM 5-HT_1B Receptor, Ki: 490 nM 5-HT_1D Receptor, Ki: 6.6 nM				5-HT₅ Receptor, Ki: 98.5 nM		Human 5-HT₇ Receptor , IC₅₀: 0.83 nM Human 5-HT₇ Receptor , Ki: 0.6 nM		99.85%
SB 258719							5-HT₇ Receptor, pKi: 7.5		99.04%
LY310762	5-HT_1D Receptor, Ki: 249 nM								98.68%
F-15599	5-HT_1A Receptor, Ki: 3.4 nM								99.82%
Tropisetron			5-HT₃ Receptor, IC₅₀: 70.1 nM						98.72%
Phenylbiguanide			5-HT₃ Receptor, EC₅₀: 3 μM						≥98.0%
JNJ-18038683							Rat 5-HT₇ Receptor, pKi: 8.19 (in HEK293 cells ) Human 5-HT₇ Receptor , pKi: 8.20 (in HEK293 cells )		99.76%
Oxatomide								serotonin	99.56%
Ecopipam hydrochloride								5-HT Receptor, Ki: 80 nM	99.46%
Rizatriptan benzoate	5-HT₁ Receptor								99.94%
Dolasetron			5-HT₃ Receptor						≥98.0%
Alverine citrate	5-HT_1A Receptor, IC₅₀: 101 nM								99.71%
(+)-Norfenfluramine		5-HT_2B Receptor, Ki: 11.2 nM 5-HT_2A Receptor, Ki: 1516 nM 5-HT_2C Receptor, Ki: 324 nM							99.92%
Xanthotoxol								serotonin	99.75%
Cyproheptadine hydrochloride sesquihydrate		5-HT₂ Receptor							99.82%
TCB2		5-HT_2A Receptor							99.21%
RU 24969	5-HT_1B Receptor, Ki: 0.38 nM 5-HT_1A Receptor, Ki: 2.5 nM								99.77%
LY 344864	human 5-HT_1F Receptor, Ki: 0.006 μM human 5-HT_1A Receptor, Ki: 0.530 μM human 5-HT_1B Receptor, Ki: 0.549 μM human 5-HT_1D Receptor, Ki: 0.575 μM human 5-HT_1E Receptor, Ki: 1.415 μM	human 5-HT_2B Receptor, Ki: 1.695 μM Human 5-HT_2A Receptor, Ki: 3.499 μM	Human 5-HT_3A Receptor, Ki: 3.935 mM				Human 5-HT₇ Receptor , Ki: 4.851 μM		98.93%
BRL 54443	5-HT_1E Receptor, Ki: 1.1 nM 5-HT_1F Receptor, Ki: 0.7 nM 5-HT_1A Receptor, Ki: 63 nM 5-HT_1B Receptor, Ki: 126 nM 5-HT_1D Receptor, Ki: 63 nM	5-HT_2A Receptor, Ki: 1259 nM 5-HT_2B Receptor, Ki: 100 nM 5-HT_2C Receptor, Ki: 316 nM				5-HT₆ Receptor, Ki: >10,000 nM	5-HT₇ Receptor, Ki: >10,000 nM		98.97%
RS-102221 hydrochloride		5-HT_2C Receptor, Ki: 10 nM							99.33%
Perospirone	5-HT_1A Receptor, Ki: 2.9 nM 5-HT₁ Receptor, Ki: 18 nM	5-HT_2A Receptor, Ki: 0.6 nM							99.43%
Ramosetron Hydrochloride			5-HT₃ Receptor						99.96%
Brilaroxazine	5-HT_1A Receptor, Ki: 1.5 nM	5-HT_2A Receptor, Ki: 2.5 nM 5-HT_2B Receptor, Ki: 0.19 nM					5-HT₇ Receptor, Ki: 2.7 nM		98.29%
Dehydroaripiprazole	5-HT_1A Receptor, Ki: 4.2 nM								99.66%
SB 243213	human 5-HT_1A Receptor, pKi: <5.3 human 5-HT_1B Receptor, pKi: 5.5 human 5-HT_1D Receptor, pKi: 6.32 human 5-HT_1E Receptor, pKi: <5.4 human 5-HT_1F Receptor, pKi: 5.35	Human 5-HT_2C Receptor, pKi: 9.37 Human 5-HT_2A Receptor, pKi: 7.01 human 5-HT_2B Receptor, pKi: 7.2				Human 5-HT₆ Receptor, pKi: 6.5	Human 5-HT₇ Receptor , pKi: 5.64		98.97%
SB 242084 dihydrochloride		5-HT_2C Receptor, pKi: 9.0							99.10%
Setiptiline		5-HT_2A Receptor 5-HT_2C Receptor	5-HT₃ Receptor						98.04%
Naftidrofuryl oxalate		5-HT₂ Receptor							98.39%
Tropisetron Hydrochloride			5-HT₃ Receptor, IC₅₀: 70.1 nM						99.97%
Flesinoxan	5-HT_1A Receptor, EC₅₀: 24 nM								99.90%
3-Hydroxy agomelatine		5-HT_2C Receptor, IC₅₀: 3.2 μM 5-HT_2C Receptor, Ki: 1.8 μM							98.00%
Opiranserin hydrochloride		5-HT_2A Receptor, IC₅₀: 1.3 μM							99.44%
(+)-Norfenfluramine hydrochloride		5-HT_2B Receptor, Ki: 11.2 nM 5-HT_2C Receptor, Ki: 324 nM 5-HT_2A Receptor, Ki: 1516 nM							99.77%
Flibanserin	5-HT_1A Receptor, Ki: 1 nM	5-HT_2A Receptor, Ki: 49 nM							99.54%
A-582941 dihydrochloride			5-HT₃ Receptor, Ki: 150 nM						99.78%
5-HT2B antagonist-1		5-HT_2B Receptor, IC₅₀: 33.4 nM							99.86%
Pizotifen		5-HT_2A Receptor							98.40%
Vabicaserin hydrochloride		5-HT_2C Receptor, EC₅₀: 8 nM							99.92%
Ocaperidone	5-HT_1A Receptor, pEC₅₀: 7.6 (h5-HT_1A) 5-HT_1A Receptor, pKi: 8.08 (h5-HT_1A)	5-HT₂ Receptor, Ki: 0.14 nM							99.93%
Geissoschizine methyl ether	5-HT_1A Receptor								99.63%
R 59-022 hydrochloride								serotonin	98.88%
Naratriptan hydrochloride	5-HT₁ Receptor								99.91%
Iloperidone	Rat 5-HT_1A Receptor, Ki: 168 nM	Rat 5-HT₂ Receptor, Ki: 3.1 nM Human 5-HT_2A Receptor, Ki: 5.6 nM Human 5-HT_2C Receptor, Ki: 42.8 nM				Rat 5-HT₆ Receptor, Ki: 42.7 μM	Rat 5-HT₇ Receptor, Ki: 21.6 nM		99.97%
Asenapine hydrochloride		5-HT_2A Receptor, Ki: 0.06 nM 5-HT_2C Receptor, Ki: 0.03 nM					5-HT₇ Receptor, Ki: 0.13 nM		99.95%
Tetrahydro-β-carboline								serotonin, Ki: 6.1 μM
NAN-190 hydrobromide	5-HT₁ Receptor								99.11%
Pumosetrag Hydrochloride			5-HT₃ Receptor						99.77%
Masupirdine mesylate						5-HT₆ Receptor, Ki: 2.04 nM			99.62%
Agomelatine hydrochloride		5-HT_2C Receptor, pKi: 6.4 (native porcine) 5-HT_2C Receptor, pKi: 6.2 (human)							99.98%
SB-399885 hydrochloride						5-HT₆ Receptor			99.58%
GR 125743	human 5-HT_1B Receptor, pKi: 8.85 human 5-HT_1D Receptor, pKi: 8.31								99.84%
Desmethyl cariprazine	5-HT_1A Receptor, Ki: 2.6 nM								98.06%
5-Carboxamidotryptamine maleate	5-HT_1A Receptor 5-HT_1B Receptor 5-HT_1D Receptor				5-HT₅ Receptor		5-HT₇ Receptor		99.73%
Deramciclane		5-HT_2A Receptor 5-HT_2C Receptor							98.13%
Mirtazapine-d₃		5-HT₂ Receptor	5-HT₃ Receptor						98.55%
Befiradol hydrochloride	5-HT_1A Receptor								99.93%
BMY 7378	5-HT_1A Receptor								99.92%
Velusetrag				5-HT₄ Receptor, pKi: 7.7					99.91%
SB 271046 Hydrochloride	5-HT_1D Receptor, pKi: 6.55 5-HT_1A Receptor, pKi: 6.35 5-HT_1B Receptor, pKi: 6.05 5-HT_1F Receptor, pKi: 5.95 5-HT_1E Receptor, pKi: <4.99	5-HT_2A Receptor, pKi: 5.62 5-HT_2B Receptor, pKi: 5.41 Human 5-HT_2C Receptor, pKi: 5.73		5-HT₄ Receptor, pKi: 5.27		5-HT₆ Receptor, pKi: 8.92-9.02	5-HT₇ Receptor, pKi: 5.39		99.93%
Urapidil hydrochloride	5-HT_1A Receptor								99.97%
VUF10166			5-HT_3A Receptor, Ki: 0.04 nM 5-HT ₃ AB, Ki: 22 nM						99.83%
Befiradol	5-HT_1A Receptor								99.20%
Methylergometrine maleate								serotonin, pA2: 9.6 nM	99.81%
Pimethixene maleate	5-HT_1A Receptor, pKi: 7.63	5-HT_2A Receptor, pKi: 10.22 5-HT_2B Receptor, pKi: 10.44 5-HT_2C Receptor, pKi: 8.42							99.94%
Flopropione	5-HT_1A Receptor								98.57%
Frovatriptan succinate hydrate	5-HT_1B Receptor, pEC₅₀: 8.2								99.60%
(Rac)-WAY-161503		5-HT_2C Receptor, Ki: 4 nM 5-HT_2C Receptor, EC₅₀: 12 nM							≥99.0%
MK-212 monohydrochloride	5-HT_1C Receptor	5-HT₂ Receptor							99.62%
Cyclobenzaprine hydrochloride		5-HT_2A Receptor							99.59%
Valerenic acid					5-HT_5A Receptor, IC₅₀: 17.2 μM				≥99.0%
WAY-181187						5-HT₆ Receptor, Ki: 2.2 nM 5-HT₆ Receptor, EC₅₀: 6.6 nM			98.07%
Intepirdine						5-HT₆ Receptor, pKi: 9.63			98.92%
Rodatristat								serotonin	99.11%
PRX-08066		5-HT_2B Receptor, IC₅₀: 3.4 nM
Nelotanserin		5-HT_2A Receptor, IC₅₀: 1.7 nM 5-HT_2C Receptor, IC₅₀: 79 nM 5-HT_2B Receptor, IC₅₀: 791 nM							99.52%
Eptapirone	5-HT_1A Receptor								99.91%
Xaliproden hydrochloride	5-HT_1A Receptor, IC₅₀: 3 nM								98.57%
RS 67333 hydrochloride				5-HT₄ Receptor, pKi: 8.7					99.73%
cis-Urocanic acid		5-HT_2A Receptor							99.92%
Eltoprazine hydrochloride	5-HT_1A Receptor 5-HT_1B Receptor	5-HT_2C Receptor							99.90%
Spiroxatrine	5-HT_1A Receptor, Ki: 3.94 nM 5-HT_1B/D Receptor, Ki: 224000 nM	5-HT₂ Receptor, Ki: 118.5 nM							99.18%
Hypidone hydrochloride	5-HT_1A Receptor								99.82%
Idalopirdine hydrochloride						5-HT₆ Receptor, Ki: 0.83 nM			99.96%
LY266097 hydrochloride		5-HT_2B Receptor, pKi: 9.8 5-HT_2A Receptor, pKi: 7.7 5-HT_2C Receptor, pKi: 7.6							99.60%
Brexpiprazole S-oxide-d₈	5-HT_1A Receptor, Ki: 0.12 nM	5-HT_2A Receptor, Ki: 0.47 nM							98.72%
Pipamperone	5-HT₁ Receptor, pKi: 5.7	5-HT_2A Receptor, pKi: 8.2 5-HT_2C Receptor, pKi: 6.9							99.89%
BMY-14802 hydrochloride	5-HT_1A Receptor								98.02%
Arotinolol		5-HT_2A Receptor							99.93%
Didesmethyl cariprazine	5-HT_1A Receptor								99.79%
Metoclopramide hydrochloride hydrate			5-HT₃ Receptor, IC₅₀: 308 nM						99.96%
LY334370	5-HT_1F Receptor, Ki: 1.6 nM								99.59%
Azasetron hydrochloride			5-HT₃ Receptor, IC₅₀: 0.33 nM						99.78%
Zolmitriptan	5-HT_1B Receptor, Ki: 5.01 nM 5-HT_1D Receptor, Ki: 0.63 nM 5-HT_1F Receptor, Ki: 63.09 nM								99.98%
DSP-1053	5-HT_1A Receptor, Ki: 5.05 nM								99.72%
Cerlapirdine						5-HT₆ Receptor			98.84%
Amperozide		5-HT_2A Receptor, Ki: 26 nM							98.75%
Piromelatine	5-HT_1A Receptor (Agonist) 5-HT_1D Receptor (Agonist)	5-HT_2B Receptor (Antagonist)							99.54%
Cyamemazine		5-HT_2A Receptor, Ki: 1.5 nM 5-HT_2C Receptor, Ki: 12 nM	5-HT₃ Receptor, Ki: 75 nM						99.42%
PU02			5-HT_3A Receptor, IC₅₀: 0.36 μM 5-HT ₃ AB, IC₅₀: 0.73 μM						≥99.0%
Cefaclor monohydrate								5-HT Receptor	99.11%
SB-200646A		5-HT_2B Receptor, pKi: 7.5 5-HT_2C Receptor, pKi: 6.9 5-HT_2A Receptor, pKi: 5.2							99.89%
(E)-3,4,5-Trimethoxycinnamic acid	5-HT_1A Receptor, IC₅₀: 7.6 μM	5-HT_2C Receptor, IC₅₀: 2.5 μM 5-HT_2A Receptor, IC₅₀: >10 μM				5-HT₆ Receptor, IC₅₀: >10 μM	5-HT₇ Receptor, IC₅₀: >10 μM		99.95%
Alniditan dihydrochloride	human 5-HT_1B Receptor, IC₅₀: 1.7 nM human 5-HT_1D Receptor, IC₅₀: 1.3 nM 5-HT_1B Receptor, Kd: 0.9 nM 5-HT_1D Receptor, Kd: 1.2 nM								99.70%
Spiramide	5-HT_1A Receptor, Ki: 50 nM 5-HT_1C Receptor, Ki: 4300 nM	5-HT₂ Receptor, Ki: 2 nM							99.23%
PRX-07034 hydrochloride	5-HT_1A Receptor, Ki: 420 nM 5-HT_1B Receptor, Ki: 260 nM 5-HT_1D Receptor, Ki: 2.8 μM	5-HT_2A Receptor, IC₅₀: 2.5 μM 5-HT_2B Receptor, IC₅₀: 2.5 μM 5-HT_2C Receptor, IC₅₀: 3.7 μM				5-HT₆ Receptor, Ki: 4-8 nM 5-HT₆ Receptor, IC₅₀: 19 nM			98.97%
YM348		5-HT_2A Receptor, Ki: 13 nM 5-HT_2B Receptor, Ki: 2.5 nM 5-HT_2C Receptor, Ki: 0.89 nM 5-HT_2A Receptor, EC₅₀: 93 nM 5-HT_2B Receptor, EC₅₀: 3.2 nM 5-HT_2C Receptor, EC₅₀: 1 nM							99.15%
RS 23597-190				5-HT₄ Receptor					99.06%
Donitriptan	5-HT_1B Receptor, pKi: 9.4 5-HT_1D Receptor, pKi: 9.3								98.06%
Renzapride				5-HT₄ Receptor, Ki: 115 nM					98.36%
RS-127445		5-HT_2B Receptor, pKi: 9.5 nM							99.62%
Bemesetron			5-HT₃ Receptor, IC₅₀: 0.33 nM						≥99.0%
p-MPPI hydrochloride	5-HT_1A Receptor								99.81%
CP-809101 hydrochloride		5-HT_2C Receptor, pEC₅₀: 9.96 5-HT_2B Receptor, pEC₅₀: 7.19 5-HT_2A Receptor, pEC₅₀: 6.81							99.37%
Isocorynoxeine		5-HT_2A Receptor, IC₅₀: 72.4 μM							99.52%
Ondansetron hydrochloride			5-HT₃ Receptor						99.94%
BRL-15572 dihydrochloride	5-HT_1D Receptor								99.77%
Ecopipam hydrobromide								5-HT Receptor, Ki: 80 nM	≥99.0%
Usmarapride free base				5-HT₄ Receptor, EC₅₀: 44 nM					99.91%
OPC-14523 hydrochloride	5-HT_1A Receptor, IC₅₀: 2.3 nM								99.95%
GSK163090	5-HT_1A Receptor, pKi: 9.4 5-HT_1B Receptor, pKi: 8.5 5-HT_1D Receptor, pKi: 9.7	5-HT_2A Receptor, pKi: 6 5-HT_2B Receptor, pKi: 6.3 5-HT_2C Receptor, pKi: 5.8				Human 5-HT₆ Receptor, pKi: <5.3	Human 5-HT₇ Receptor , pKi: 6.8		99.77%
GR-46611	5-HT_1D Receptor								99.82%
Adoprazine	5-HT_1A Receptor, pEC₅₀: 9 5-HT_1A Receptor, pKi: 9.1						5-HT₇ Receptor, pKi: 7.2		98.60%
Strictosidinic acid								5-HT Receptor
Iferanserin		5-HT_2A Receptor							99.74%
Temanogrel		5-HT_2A Receptor, Ki: 4.9 nM							98.14%
Ampreloxetine								5-HT Receptor	98.49%
E-3620			5-HT₃ Receptor						98.88%
Urapidil	5-HT_1A Receptor								99.30%
Nemonapride	5-HT_1A Receptor, IC₅₀: 34 nM								99.90%
Flumexadol		5-HT_2C Receptor, Ki: 25 nM							99.86%
ST1936		5-HT_2B Receptor, Ki: 245 nM				5-HT₆ Receptor, Ki: 13 nM	5-HT₇ Receptor, Ki: 168 nM		99.70%
Velusetrag hydrochloride				5-HT₄ Receptor, pKi: 7.7					98.95%
Perospirone hydrochloride	5-HT_1A Receptor, Ki: 2.9 nM 5-HT₁ Receptor, Ki: 18 nM	5-HT_2A Receptor, Ki: 0.6 nM							99.94%
TC-2153	5-HT_1A Receptor	5-HT_2A Receptor							98.73%
WAY-100135 dihydrochloride	5-HT_1A Receptor, IC₅₀: 34 nM								98.32%
Felcisetrag				huamn 5-HT_4(c) Receptor, pKi: 9.4					99.94%
SB-616234-A	5-HT_1B Receptor								98.14%
Aripiprazole-d₈		5-HT_2A Receptor 5-HT_2C Receptor							≥99.0%
Almotriptan malate	5-HT_1B Receptor 5-HT_1D Receptor								99.53%
Naronapride				5-HT₄ Receptor					99.79%
Indophagolin						5-HT₆ Receptor, IC₅₀: 1.0 μM			98.05%
UNC9994	5-HT_1F Receptor, Ki: 26 nM	5-HT_2A Receptor, Ki: 140 nM 5-HT_2B Receptor, Ki: 25 nM 5-HT_2C Receptor, Ki: 512 nM							98.06%
Ro60-0175		5-HT_2C Receptor							99.98%
Org-12962		5-HT_2C Receptor, pEC₅₀: 7.01 5-HT_2A Receptor, pEC₅₀: 6.38 5-HT_2B Receptor, pEC₅₀: 6.28							99.93%
LY-272015 hydrochloride		5-HT_2B Receptor							99.54%
Pizotifen malate		5-HT_2A Receptor							99.88%
AVN-492						5-HT₆ Receptor, Ki: 91 pM			99.30%
Mosapride citrate dihydrate				5-HT₄ Receptor
Usmarapride				5-HT₄ Receptor, EC₅₀: 44 nM					≥98.0%
Rodatristat ethyl	5-HT₁ Receptor								≥98.0%
5-Methoxytryptamine hydrochloride	5-HT₁ Receptor	5-HT₂ Receptor		5-HT₄ Receptor	5-HT₅ Receptor	5-HT₆ Receptor	5-HT₇ Receptor		≥98.0%
LE 300		Rat 5-HT_2A, pA2: 8.32							98.5%
Cariprazine-d₆	5-HT_1A Receptor, Ki: 2.6 nM								98.00%
PNU-142633	5-HT_1D Receptor, Ki: 6 nM								98.6%
Peptide 401								serotonin	98.26%
Pruvanserin		5-HT_2A Receptor							99.27%
SB 243213 dihydrochloride	human 5-HT_1A Receptor, pKi: <5.3 human 5-HT_1B Receptor, pKi: 5.5 human 5-HT_1D Receptor, pKi: 6.32 human 5-HT_1E Receptor, pKi: <5.4 human 5-HT_1F Receptor, pKi: 5.35	Human 5-HT_2C Receptor, pKi: 9.37 Human 5-HT_2A Receptor, pKi: 7.01 human 5-HT_2B Receptor, pKi: 7.2				Human 5-HT₆ Receptor, pKi: 6.5	Human 5-HT₇ Receptor , pKi: 5.64		≥99.0%
Eplivanserin hemifumarate		5-HT_2A Receptor, IC₅₀: 5.8 nM 5-HT_2C Receptor, IC₅₀: 120 nM							98.07%
Cinanserin hydrochloride		5-HT₂ Receptor, Ki: 41 nM							99.48%
Repinotan	5-HT_1A Receptor, Ki: 0.19 nM (In calf hippocampus) 5-HT_1A Receptor, Ki: 0.25 nM (In rat and human cortex) 5-HT_1A Receptor, Ki: 0.59 nM (In rat hippocampus)						5-HT₇ Receptor, Ki: 6 nM
F 13714 fumarate	5-HT_1A Receptor								99.05%
SB-216641A	5-HT_1B Receptor 5-HT_1D Receptor								≥98.0%
GR127935 hydrochloride	5-HT_1B Receptor, pKi: 8.5 5-HT_1D Receptor, pIC₅₀: 8.5								98.1%
Spiperone hydrochloride	5-HT_1A Receptor, Ki: 49 nM	5-HT_2A Receptor, Ki: 1 nM							99.10%
AP521	5-HT_1A Receptor, IC₅₀: 94 nM (in human) 5-HT_1A Receptor, IC₅₀: 135 nM (in rat) 5-HT_1B Receptor, IC₅₀: 254 nM (in rat) 5-HT_1B Receptor, IC₅₀: 5530 nM (in human) 5-HT_1D Receptor, IC₅₀: 418 nM (in human)				5-HT_5A Receptor, IC₅₀: 422 nM (in human)		5-HT₇ Receptor, IC₅₀: 198 nM (in rat)		98.96%
Facinicline hydrochloride			5-HT₃ Receptor, Ki: 1.2 nM						99.93%
NPS ALX Compound 4a						5-HT₆ Receptor, IC₅₀: 7.2 nM 5-HT₆ Receptor, Ki: 0.2 nM			≥99.0%
4F 4PP oxalate		5-HT_2A Receptor, Ki: 5.3 nM 5-HT_2C Receptor, Ki: 620 nM							98.08%
SB228357		5-HT_2A Receptor, pKi: 6.9 5-HT_2C Receptor, pKi: 9 5-HT_2B Receptor, pKi: 8							99.43%
(R)-Mirtazapine			5-HT₃ Receptor						99.79%
RS 39604				5-HT₄ Receptor, pKi: 9.1					≥98.0%
PF-04995274				5-HT₄ Receptor					99.95%
5-HT1A modulator 1		5-HT_2A Receptor, IC₅₀: 500 nM 5-HT_2C Receptor, IC₅₀: 4000 nM
Ipsapirone	5-HT_1A Receptor								99.87%
EMD 56551	5-HT_1A Receptor
FPT	5-HT_1A Receptor, IC₅₀: 39.3 nM 5-HT_1B Receptor, IC₅₀: 1.2 nM 5-HT_1D Receptor, IC₅₀: 0.5 nM 5-HT_1A Receptor, Ki: 4.3 nM 5-HT_1B Receptor, Ki: 2.3 nM 5-HT_1D Receptor, Ki: 1.2 nM 5-HT_1F Receptor, Ki: >10,000 nM								98.06%
S-14506 hydrochloride	5-HT₁ Receptor	5-HT_2A Receptor 5-HT_2C Receptor							99.92%
Fananserin		5-HT₂ Receptor, Ki: 0.37 nM							99.97%
(S)-Amisulpride							5-HT₇ Receptor, Ki: 900 nM		99.75%
SKF-83566 hydrobromide		5-HT₂ Receptor, Ki: 11 nM
Fabesetron			5-HT₃ Receptor	5-HT₄ Receptor
(R)-Praziquantel-d₁₁		5-HT_2B Receptor							99.57%
BIMU 8				5-HT₄ Receptor, EC₅₀: 18 nM					≥99.0%
cis-(Z)-Flupentixol dihydrochloride		5-HT_2A Receptor, Ki: 7 nM
OPC-14523 free base	5-HT_1A Receptor, IC₅₀: 2.3 nM
5-HT2A antagonist 1		5-HT_2A Receptor
Ro60-0175 fumarate		5-HT_2C Receptor							99.47%
Lecozotan hydrochloride	5-HT_1A Receptor, Ki: 4.5 nM								98.71%
Almotriptan	5-HT_1B Receptor 5-HT_1D Receptor								99.94%
Brexpiprazole S-oxide	5-HT_1A Receptor, Ki: 0.12 nM	5-HT_2A Receptor, Ki: 0.47 nM
BMY 14802	5-HT_1A Receptor								98.96%
SB 243213 hydrochloride	human 5-HT_1A Receptor, pKi: <5.3 human 5-HT_1B Receptor, pKi: 5.5 human 5-HT_1D Receptor, pKi: 6.32 human 5-HT_1E Receptor, pKi: <5.4 human 5-HT_1F Receptor, pKi: 5.35	Human 5-HT_2C Receptor, pKi: 9.37 Human 5-HT_2A Receptor, pKi: 7.01 human 5-HT_2B Receptor, pKi: 7.2				Human 5-HT₆ Receptor, pKi: 6.5	Human 5-HT₇ Receptor , pKi: 5.64
Lesopitron dihydrochloride	5-HT_1A Receptor, IC₅₀: 125 nM (in rat hippocampal membranes)								≥98.0%
Tedatioxetine hydrobromide		5-HT_2A Receptor 5-HT_2C Receptor	5-HT₃ Receptor						99.83%
Naluzotan	5-HT_1A Receptor, IC₅₀: 20 nM 5-HT_1A Receptor, Ki: 5.1 nM								98.05%
Relenopride hydrochloride		5-HT_2A Receptor, Ki: 600 nM 5-HT_2B Receptor, Ki: 31 nM 5-HT_2B Receptor, IC₅₀: 2.1 μM		5-HT₄ Receptor, Ki: 4.96 nM					99.85%
Flibanserin hydrochloride (propan-2-ol) hydrate	5-HT_1A Receptor, Ki: 1 nM	5-HT_2A Receptor, Ki: 49 nM							99.04%
Eplivanserin (mixture)		5-HT_2A Receptor							99.77%
Isopteropodine		5-HT₂ Receptor							98.66%
MAO-A/5-HT2AR-IN-1		5-HT_2A Receptor, IC₅₀: 0.014 μM							99.71%
CJ033466				5-HT₄ Receptor, EC₅₀: 9 nM					98.29%
LY 344864 racemate	5-HT_1F Receptor								98.07%
(S)-Mirtazapine		5-HT₂ Receptor	5-HT₃ Receptor						99.76%
ARC 239	5-HT_1A Receptor, Ki: 63.1 nM								99.71%
Risperidone hydrochloride		5-HT₂ Receptor, Ki: 4.8 nM
(Rac)-Rotigotine hydrochloride	5-HT_1A Receptor, Ki: 30 nM	5-HT_2B Receptor, Ki: 27 nM							98.66%
Dolasetron Mesylate hydrate			5-HT₃ Receptor						≥99.0%
Alosetron			5-HT₃ Receptor
Mosapride				5-HT₄ Receptor
(-)-5-HT2C agonist-3		5-HT_2A Receptor, IC₅₀: 72 nM 5-HT_2C Receptor, IC₅₀: 103 nM 5-HT_2B Receptor, IC₅₀: 570 nM
Pardoprunox hydrochloride	5-HT_1A Receptor, pEC₅₀: 6.3								99.46%
Eltoprazine	5-HT_1A Receptor 5-HT_1B Receptor	5-HT_2C Receptor
Pimethixene	5-HT_1A Receptor, pKi: 7.63	5-HT_2A Receptor, pKi: 10.22 5-HT_2B Receptor, pKi: 10.44 5-HT_2C Receptor, pKi: 8.42
Ziprasidone hydrochloride	Rat 5-HT_1A Receptor, Ki: 3.4 nM	Rat 5-HT_2A, Ki: 0.42 nM
Palonosetron			5-HT₃ Receptor
Viloxazine		Human 5-HT_2C Receptor, EC₅₀: 32 μM human 5-HT_2B Receptor, IC₅₀: 27 μM
Cyanopindolol	5-HT_1A Receptor, Ki: 2.1 nM 5-HT_1B Receptor, Ki: 3 nM
5-HT6/7 antagonist 1		5-HT_2A Receptor				5-HT₆ Receptor	5-HT₇ Receptor
Revexepride				5-HT₄ Receptor					99.84%
Lintopride			5-HT₃ Receptor	5-HT₄ Receptor
Naratriptan	5-HT₁ Receptor
(±)-Fabesetron hydrochloride			5-HT₃ Receptor	5-HT₄ Receptor
Lidanserin		5-HT_2A Receptor							≥98.0%
SB-269970							Human 5-HT₇ Receptor , pKi: 8.3
SEP-363856	5-HT_1A Receptor, EC₅₀: 2.3 μM 5-HT_1B Receptor, EC₅₀: 15.6 μM 5-HT_1D Receptor, EC₅₀: 0.262 μM	5-HT_2A Receptor, EC₅₀: >10 μM 5-HT_2C Receptor, EC₅₀: 30 μM					5-HT₇ Receptor, EC₅₀: 6.7 μM
Clocapramine		5-HT_2A Receptor
CYB210010	5-HT_1A Receptor, Ki: 32 nM 5-HT_1B Receptor, Ki: 949 nM	5-HT_2A Receptor, EC₅₀: 4.1 nM 5-HT_2C Receptor, EC₅₀: 7.3 nM 5-HT_2B Receptor, EC₅₀: 88 nM				5-HT₆ Receptor, Ki: 1301 nM	5-HT₇ Receptor, Ki: 4918 nM
LY334370 hydrochloride	5-HT_1F Receptor, Kd: 0.446 nM
UCSF648					5-HT_5A Receptor
Blonanserin dihydrochloride		5-HT_2A Receptor, Ki: 0.812 nM 5-HT_2C Receptor, Ki: 26.4 nM				5-HT₆ Receptor, Ki: 11.7 nM
SB 271046						5-HT₆ Receptor, pKi: 8.92-9.09
Scopolamine hydrochloride			5-HT₃ Receptor, IC₅₀: 2.09 μM
Metoclopramide hydrochloride			5-HT₃ Receptor, IC₅₀: 308 nM
5-HT7 receptor ligand 1							5-HT₇ Receptor, Ki: 8 nM
Opiranserin		5-HT_2A Receptor, IC₅₀: 1.3 μM
Isamoltane hemifumarate	5-HT_1B Receptor, IC₅₀: 39 nM
WAY-181187 oxalate						5-HT₆ Receptor, Ki: 2.2 nM 5-HT₆ Receptor, EC₅₀: 6.6 nM
BRL-15572 hydrochloride	5-HT_1D Receptor
Mesulergine hydrochloride		5-HT_2C Receptor
5-HT2CR agonist 1		5-HT_2C Receptor, EC₅₀: 121.5 nM
Capeserod				5-HT₄ Receptor, Ki: 0.6 nM
Remlifanserin		5-HT_2A Receptor
Methylergometrine		5-HT_2B Receptor
Blonanserin-d₈		5-HT₂ Receptor
MM 77 dihydrochloride	5-HT_1A Receptor
ZINC866533340		5-HT_2A Receptor, Ki: 1.6 nM
RS-102221		5-HT_2C Receptor, Ki: 10 nM
VU6067416		5-HT_2A Receptor, EC₅₀: 189 nM
CART(62-76)(human,rat) TFA								serotonin
Dehydro Palonosetron			5-HT₃ Receptor
5-HT2A antagonist 2		5-HT_2A Receptor, IC₅₀: 14 nM
Donitriptan hydrochloride	5-HT_1B Receptor, pKi: 9.4 5-HT_1D Receptor, pKi: 9.3
NPS ALX Compound 4a dihydrochloride						5-HT₆ Receptor, IC₅₀: 7.2 nM 5-HT₆ Receptor, Ki: 0.2 nM
5-HT6/5-HT2A receptor ligand-2		5-HT_2A Receptor, Ki: 32 nM				5-HT₆ Receptor, Ki: 25 nM
Cisapride monohydrate				5-HT₄ Receptor, EC₅₀: 0.14 μM
BMY 28674	Rat 5-HT_1A Receptor, EC₅₀: 4 μM Rat 5-HT_1A Receptor, EC₅₀: 1 μM
GSK215083						5-HT₆ Receptor
5-HT3 antagonist 5			5-HT₃ Receptor						99.75%
3-AQC			5-HT₃ Receptor
S-14671	5-HT_1A Receptor, pKi: 9.3
MAO-B-IN-3						Human 5-HT₆ Receptor, Ki: 696 nM
Tandospirone hydrochloride	5-HT_1A Receptor, Ki: 27 nM
Brexpiprazole hydrochloride	5-HT_1A Receptor, Ki: 0.12 nM	5-HT_2A Receptor, Ki: 0.47 nM
SB 258719 hydrochloride							5-HT₇ Receptor, pKi: 7.5
(R)-Mirtazapine-d₃			5-HT₃ Receptor
LY320135		5-HT₂ Receptor, Ki: 6.4 μM
DU125530	5-HT_1A Receptor, Ki: 0.7 nM 5-HT_1B Receptor, Ki: 890 nM 5-HT_1C Receptor, Ki: 1200 nM	5-HT_2A Receptor, Ki: 240 nM 5-HT_2C Receptor, Ki: 750 nM	5-HT₃ Receptor, Ki: 1100 nM
Org-12962 hydrochloride		5-HT_2C Receptor, pEC₅₀: 7.01 5-HT_2A Receptor, pEC₅₀: 6.38 5-HT_2B Receptor, pEC₅₀: 6.28
Perphenazine dihydrochloride	5-HT_1A Receptor, Ki: 421 nM	5-HT_2A Receptor, Ki: 5.6 nM 5-HT_2C Receptor, Ki: 132 nM				5-HT₆ Receptor, Ki: 17 nM	5-HT₇ Receptor, Ki: 23 nM
Urapidil-d₄	5-HT_1A Receptor
AVN-101 hydrochloride	5-HT_1B Receptor, Ki: 720 nM 5-HT_1A Receptor, Ki: 61 nM	5-HT_2A Receptor, Ki: 1.56 nM 5-HT_2C Receptor, Ki: 1.17 nM 5-HT_2B Receptor, Ki: 10.6 nM				5-HT₆ Receptor, Ki: 2.04 nM	5-HT₇ Receptor, Ki: 0.153 nM		99.59%
SUN C5174		5-HT₂ Receptor
Asenapine citrate	5-HT_1B Receptor, pKi: 8.4 5-HT_1A Receptor, pKi: 8.6	5-HT_2A Receptor, pKi: 10.2 5-HT_2C Receptor, pKi: 10.5 5-HT_2B Receptor, pKi: 9.8			5-HT₅ Receptor, pKi: 8.8	5-HT₆ Receptor, pKi: 9.6	5-HT₇ Receptor, pKi: 9.9
2-Methyl-5-HT hydrochloride			5-HT₃ Receptor
PNU-282987 free base			5-HT₃ Receptor
BGC20-761		Human 5-HT_2A Receptor, Ki: 69 nM				Human 5-HT₆ Receptor, Ki: 20 nM
Robalzotan	5-HT_1A Receptor
Ro 04-6790						Rat 5-HT₆ Receptor, pKi: 7.26 Human 5-HT₆ Receptor, pKi: 7.35
SB-200646		5-HT_2B Receptor, pKi: 7.5 5-HT_2C Receptor, pKi: 6.9 5-HT_2A Receptor, pKi: 5.2
Risperidone-d₆		5-HT_2A Receptor, Ki: 4.8 nM
RU 24969 hemisuccinate	5-HT_1A Receptor, Ki: 2.5 nM 5-HT_1B Receptor, Ki: 0.38 nM
Frovatriptan succinate	5-HT_1B Receptor, pEC₅₀: 8.2
5-HT6/5-HT2AR antagonist-1		5-HT_2A Receptor, Ki: 39 nM				5-HT₆ Receptor, Ki: 11 nM
Lurosetron			5-HT₃ Receptor
F 13714	5-HT_1A Receptor, pKi: 10.23 5-HT_1B Receptor, pIC₅₀: 5.12
LY 278584			5-HT₃ Receptor, Ki: 1.62 nM
SB-221284		5-HT_2A Receptor, pKi: 6.4 5-HT_2B Receptor, pKi: 7.9 5-HT_2C Receptor, pKi: 8.6
SCH-23390 maleate		5-HT_2C Receptor, Ki: 9.3 nM
GR127935	5-HT_1D Receptor
NAN-190	5-HT₁ Receptor
SEP-363856 mesylate	5-HT_1A Receptor, EC₅₀: 2.3 μM 5-HT_1B Receptor, EC₅₀: 15.6 μM 5-HT_1D Receptor, EC₅₀: 0.262 μM	5-HT_2A Receptor, EC₅₀: >10 μM 5-HT_2C Receptor, EC₅₀: 30 μM					5-HT₇ Receptor, EC₅₀: 6.7 μM
(Rac)-WAY-161503 hydrochloride		5-HT_2C Receptor, Ki: 4 nM 5-HT_2C Receptor, EC₅₀: 12 nM
(+)-Norcisapride			5-HT₃ Receptor	5-HT₄ Receptor
SB-215505		5-HT_2B Receptor, pKi: 8.3 5-HT_2A Receptor, pKi: 6.77 5-HT_2C Receptor, pKi: 7.66							98.91%
Sumatriptan hydrochloride	5-HT_1D Receptor, Ki: 17 nM 5-HT_1B Receptor, Ki: 27 nM 5-HT_1A Receptor, Ki: 100 nM 5-HT_1D Receptor, IC₅₀: 7.3 nM 5-HT_1B Receptor, IC₅₀: 9.3 nM 5-HT_1F Receptor, IC₅₀: 17.8 nM
EMD386088						5-HT₆ Receptor			99.06%
SB399885						5-HT₆ Receptor, pKi: 9.02 Human 5-HT₆ Receptor, pKi: 9.11
Cinitapride monotartrate	5-HT₁ Receptor	5-HT₂ Receptor		5-HT₄ Receptor
Ziprasidone mesylate	Rat 5-HT_1A Receptor, Ki: 3.4 nM	Rat 5-HT₂ Receptor, Ki: 0.42 nM
MK-212	5-HT_1C Receptor	5-HT₂ Receptor
Robalzotan hydrochloride	5-HT_1A Receptor								99.5%
1-(1-Naphthyl)piperazine hydrochloride	5-HT_1A Receptor	5-HT_2A Receptor
SB 258741 hydrochloride							5-HT₇ Receptor
SGS518 oxalate						5-HT₆ Receptor
Trimipramine	5-HT_1C Receptor, pKi: 6.39 5-HT_1A Receptor, pKi: 4.66	5-HT₂ Receptor, pKi: 8.10
ST1936 oxalate		5-HT_2B Receptor, Ki: 245 nM				5-HT₆ Receptor, Ki: 13 nM	Human 5-HT₇ Receptor , Ki: 168 nM
LY215840		5-HT₂ Receptor					5-HT₇ Receptor
Masupirdine free base						5-HT₆ Receptor, Ki: 2.04 nM
Sarpogrelate		5-HT₂ Receptor
ML 10302 hydrochloride			5-HT₃ Receptor, Ki: 782 nM	5-HT₄ Receptor, EC₅₀: 4 nM 5-HT₄ Receptor, Ki: 1.07 nM
GM-60186		5-HT_2B Receptor, IC₅₀: 257 nM
5-HT6R antagonist 3	5-HT_1A Receptor, Ki: 3533 nM	5-HT_2A Receptor, Ki: 35 nM				5-HT₆ Receptor, Ki: 14 nM	5-HT₇ Receptor, Ki: 1449 nM
Syk Inhibitor II hydrochloride								5-HT Receptor, IC₅₀: 460 nM
Piclozotan	5-HT_1A Receptor
Mesembrine								serotonin, Ki: 1.4 nM
SB-737050A						5-HT₆ Receptor
U92016A hydrochloride	5-HT_1A Receptor, Ki: 0.2 nM
Blonanserin-d₅		5-HT₂ Receptor
Aripiprazole monohydrate	5-HT_1A Receptor	5-HT_2A Receptor 5-HT_2B Receptor 5-HT_2C Receptor
CART(62-76)(human,rat)								serotonin
DR4485 hydrochloride							5-HT₇ Receptor, pKi: 8.14
Syk Inhibitor II dihydrochloride								5-HT Receptor, IC₅₀: 460 nM
WAY-181187 hydrochloride						5-HT₆ Receptor, Ki: 2.2 nM 5-HT₆ Receptor, EC₅₀: 6.6 nM
LY320954		5-HT_2A Receptor, Ki: 96 nM 5-HT_2B Receptor, Ki: 1642 nM 5-HT_2C Receptor, Ki: 257 nM
5-HT6R/MAO-B modulator 1						5-HT₆ Receptor
TIK-301		5-HT_2C Receptor 5-HT_2B Receptor
EMDT oxalate						5-HT₆ Receptor
WAY 629		5-HT_2C Receptor, EC₅₀: 426 nM 5-HT_2A Receptor, EC₅₀: 260000 nM
Ziprasidone mesylate trihydrate	Rat 5-HT_1A Receptor, Ki: 3.4 nM	Rat 5-HT₂ Receptor, Ki: 0.42 nM
PRX-08066 maleate		5-HT_2B Receptor, IC₅₀: 3.4 nM
LP 12 hydrochloride	5-HT_1A Receptor, IC₅₀: 60.9 nM	5-HT_2A Receptor, IC₅₀: 1464 nM					5-HT₇ Receptor, IC₅₀: 0.13 nM
Asimilobine								serotonergic receptor
5-HT7R antagonist 2							5-HT₇ Receptor, Ki: 67 nM
RS-64459-193	5-HT_1A Receptor, Ki: 24.9 nM (CHO cells) human 5-HT_1A Receptor, pKi: 7.6 (Sf9) human 5-HT_1A Receptor, pKi: 7.04	5-HT_2C Receptor, pKi: 6.87 Rat 5-HT_2A, pKi: 7.02	5-HT₃ Receptor, pKi: <4				Human 5-HT₇ Receptor , pKi: 7.18
5-HT1A antagonist 1	5-HT_1A Receptor, Ki: 35 nM	5-HT_2A Receptor, Ki: 530 nM					5-HT₇ Receptor, Ki: 462 nM
PF-4479745	5-HT_1A Receptor, IC₅₀: 500 nM	5-HT_2C Receptor, EC₅₀: 10 nM 5-HT_2C Receptor, Ki: 15 nM 5-HT_2A Receptor, IC₅₀: 360 nM 5-HT_2B Receptor, IC₅₀: 67 nM				5-HT₆ Receptor, IC₅₀: 280 nM
2-Methyl-5-HT maleate			5-HT₃ Receptor
NEO 376	5-HT₁ Receptor								99.23%
CP 93129	5-HT_1B Receptor
Loxapine hydrochloride		human 5-HT₂
E6801						5-HT₆ Receptor
Lintopride hydrochloride			5-HT₃ Receptor	5-HT₄ Receptor
5HT6-ligand-2						5-HT₆ Receptor
MR33317				5-HT₄ Receptor
3-Hydroxy agomelatine-d₃		5-HT_2C Receptor, IC₅₀: 3.2 μM 5-HT_2C Receptor, Ki: 1.8 μM							99.92%
7-Desmethyl-3-hydroxyagomelatine		5-HT_2C Receptor
5-Carboxamidotryptamine	5-HT_1A Receptor 5-HT_1B Receptor 5-HT_1D Receptor				5-HT_5A Receptor		5-HT₇ Receptor
Bifeprunox	5-HT_1A Receptor, pKi: 7.19 (cortex) 5-HT_1A Receptor, pEC₅₀: 6.37 (hippocampus)
Dehydroaripiprazole hydrochloride	5-HT_1A Receptor, Ki: 4.2 nM
CP-135807	5-HT_1D Receptor, IC₅₀: 3.1 nM (rat) 5-HT_1D Receptor, IC₅₀: 33 nM (bovine)
Antipsychotic agent-2	5-HT_1A Receptor, EC₅₀: 160 nM	5-HT_2A Receptor, Kb: 96.4 nM
Syk Inhibitor II dihydrochloride dihydrate								serotonin, IC₅₀: 460 nM
5-HT6/5-HT2A receptor ligand-1		5-HT_2A Receptor, IC₅₀: 11 nM				5-HT₆ Receptor, Ki: 2 nM
WAY 629 hydrochloride		5-HT_2C Receptor, EC₅₀: 426 nM 5-HT_2A Receptor, EC₅₀: 260000 nM
DSP-1053 benzenesulfonate	5-HT_1A Receptor, Ki: 5.05 nM
Carpindolol	5-HT_1B Receptor, pKd: 8.53 5-HT_1D Receptor, pEC₅₀: 5.91 5-HT_1D Receptor, pKd: 6.37
DV-7028 hydrochloride		5-HT₂ Receptor
PNU-96415E		5-HT_2A Receptor
Ecopipam								5-HT Receptor, Ki: 80 nM
PF-03382792				5-HT_4d Receptor, Ki: 2.7 nM 5-HT_4d Receptor, EC₅₀: 0.9 nM
Eletriptan	5-HT_1B Receptor, pKi: 8.0 5-HT_1D Receptor, pKi: 8.9
CP94253	5-HT_1B Receptor, Ki: 2 nM 5-HT_1D Receptor, Ki: 49 nM 5-HT_1A Receptor, Ki: 89 nM 5-HT_1C Receptor, Ki: 860 nM	5-HT₂ Receptor, Ki: 1600 nM
BL-1020 mesylate		5-HT_2A Receptor, Ki: 3.74 μM
PF-03246799		5-HT_2C Receptor, EC₅₀: 190 nM 5-HT_2C Receptor, Ki: 160 nM
Capeserod hydrochloride				5-HT_4(e) Receptor, Ki: 0.6 nM
Itasetron			5-HT₃ Receptor
WAY-100289			5-HT₃ Receptor
SB-272183	5-HT_1A Receptor, pKi: 8.0 5-HT_1B Receptor, pKi: 8.1 5-HT_1D Receptor, pKi: 8.7
EGIS-7625		5-HT_2B Receptor, pKi: 9.0 5-HT_2A Receptor, pKi: 6.2 5-HT_2C Receptor, pKi: 7.7
(R)-Praziquantel		5-HT_2B Receptor
VER-3323		Human 5-HT_2C Receptor
Risperidone mesylate		5-HT_2A Receptor, Ki: 4.8 nM
MS 245						5-HT₆ Receptor, Ki: 1.5 nM
PD 118717	5-HT₁ Receptor
PF-05212377						Human 5-HT₆ Receptor
DA-6886 monohydrochloride				5-HT₄ Receptor, pIC₅₀: 4.3
Iloperidone hydrochloride	Rat 5-HT_1A Receptor, Ki: 168 nM	Rat 5-HT₂ Receptor, Ki: 3.1 nM Human 5-HT_2A Receptor, Ki: 5.6 nM Human 5-HT_2C Receptor, Ki: 42.8 nM				Rat 5-HT₆ Receptor, Ki: 42.7 nM	Rat 5-HT₇ Receptor, Ki: 21.6 nM
Cinanserin	5-HT₁ Receptor, Ki: 3500 nM	5-HT₂ Receptor, Ki: 41 nM
Agomelatine (L(+)-Tartaric acid)		5-HT_2C Receptor, pKi: 6.4 (native porcine) 5-HT_2C Receptor, pKi: 6.2 (human)							99.82%
SC-53116				5-HT₄ Receptor, EC₅₀: 23 nM
Cloroperone		human 5-HT₂, Ki: 4.5 nM
Alosetron ((Z)-2-butenedioate)			5-HT₃ Receptor
Ro 63-0563						Rat 5-HT₆ Receptor, pKi: 7.83 Human 5-HT₆ Receptor, pKi: 7.91
Zalospirone	5-HT_1A Receptor
Beloxepin		5-HT₂ Receptor
Pardoprunox	5-HT_1A Receptor, pEC₅₀: 6.3
Dolasetron Mesylate			5-HT₃ Receptor
Serazapine		5-HT₂ Receptor
Alosetron (Hydrochloride(1:X))			5-HT₃ Receptor
S14063	5-HT_1A Receptor
Sarizotan dihydrochloride	5-HT_1A Receptor, IC₅₀: 0.1 nM	5-HT_2A Receptor, IC₅₀: 587 nM 5-HT_2B Receptor, IC₅₀: 108 nM			5-HT_5A Receptor, IC₅₀: 313 nM	Human 5-HT₆ Receptor, IC₅₀: 3300 nM	Human 5-HT₇ Receptor , IC₅₀: 10 nM
Idalopirdine						5-HT₆ Receptor, Ki: 0.83 nM
R(+)-8-OH-DPAT hydrobromide	5-HT_1A Receptor
GTS-21			5-HT_3A Receptor, IC₅₀: 3.1 μM
Etoperidone hydrochloride	5-HT_1A Receptor, Kd: 85 nM	5-HT₂ Receptor, Kd: 36 nM
Piboserod hydrochloride				5-HT₄ Receptor
Fabesetron hydrochloride			5-HT₃ Receptor	5-HT₄ Receptor
Nexopamil racemate		5-HT₂ Receptor
Abaperidone		5-HT_2A Receptor, IC₅₀: 6.2 nM
Irindalone		5-HT₂ Receptor
Pancopride			5-HT₃ Receptor
Sulamserod				5-HT₄ Receptor
Alniditan	human 5-HT_1B Receptor, IC₅₀: 1.7 nM (in HEK 293 cell) human 5-HT_1D Receptor, IC₅₀: 1.3 nM (in HEK 293 cell) 5-HT_1B Receptor, Kd: 0.9 nM 5-HT_1D Receptor, Kd: 1.2 nM
RG-12915			5-HT₃ Receptor, IC₅₀: 0.16 nM
NRA-0160		5-HT_2A Receptor, Ki: 180 nM (in rat)
MHP 133				5-HT₄ Receptor
Wf-516	5-HT_1A Receptor, Ki: 5 nM	5-HT_2A Receptor, Ki: 40 nM
T 82			5-HT₃ Receptor
Clozapine hydrochloride		5-HT_2A Receptor, Ki: 4 nM
CP-809101		5-HT_2C Receptor, pEC₅₀: 9.96 5-HT_2B Receptor, pEC₅₀: 7.19 5-HT_2A Receptor, pEC₅₀: 6.81
Adatanserin	5-HT_1A Receptor, Ki: 1 nM	5-HT₂ Receptor, Ki: 73 nM
CGS 12066 dimaleate	5-HT_1B Receptor, IC₅₀: 51 nM
AM9405			5-HT₃ Receptor, IC₅₀: 0.076 nM
Clocapramine dihydrochloride hydrate		5-HT_2A Receptor
5-HT7 agonist 1							5-HT₇ Receptor
WAY 163909		5-HT_2C Receptor, Ki: 10.5±1.1 nM
PRX933 hydrochloride		5-HT_2C Receptor
Eplivanserin		5-HT_2A Receptor, IC₅₀: 5.8 nM (in rat cortical membrane) 5-HT_2A Receptor, Ki: 1.14 nM 5-HT_2C Receptor, IC₅₀: 120 nM
5-HT4 antagonist 1				5-HT₄ Receptor, pKi: 9.6					98.67%
5-HT3 antagonist 3			5-HT₃ Receptor, Ki: 0.25 nM
AR-A 2	5-HT_1A Receptor, Ki: 3070 nM 5-HT_1B/D Receptor, Ki: 20 nM	5-HT_2A Receptor, Ki: 339 nM
LY 344864 hydrochloride	human 5-HT_1F Receptor, Ki: 0.006 μM human 5-HT_1A Receptor, Ki: 0.530 μM human 5-HT_1B Receptor, Ki: 0.549 μM human 5-HT_1D Receptor, Ki: 0.575 μM human 5-HT_1E Receptor, Ki: 1.415 μM	human 5-HT_2B Receptor, Ki: 1.695 μM Human 5-HT_2C Receptor, Ki: 3.499 μM	Human 5-HT_3A Receptor, Ki: 3.935 μM				Human 5-HT₇ Receptor , Ki: 4.851 μM
Zatosetron maleate			5-HT₃ Receptor
(4E)-SUN9221		5-HT₂ Receptor
5-HT3 antagonist 1			5-HT₃ Receptor
5-HT3-In-1			5-HT₃ Receptor
5-HT2 antagonist 1		5-HT₂ Receptor
5-HT3 antagonist 2			5-HT₃ Receptor
5HT6-ligand-1						5-HT₆ Receptor, Ki: 1.43 nM

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